TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Binding affinity to HRAS (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of HRAS (unknown origin) farnesylationMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human H-rasMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Tested for 50% inhibition of generation of Human Ha-ras polymerase chain reaction(PCR) productsMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Tested for 50% inhibition of generation of Human Ha-ras polymerase chain reaction(PCR) productsMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Tested for 50% inhibition of generation of Human Ha-ras polymerase chain reaction(PCR) productsMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Tested for 50% inhibition of generation of Human Ha-ras polymerase chain reaction(PCR) productsMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Tested for 50% inhibition of generation of Human Ha-ras polymerase chain reaction(PCR) productsMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Tested for 50% inhibition of generation of Human Ha-ras polymerase chain reaction(PCR) productsMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Tested for 50% inhibition of generation of Human Ha-ras polymerase chain reaction(PCR) productsMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 88nMAssay Description:Concentration required to inhibit 50% of the cultured colonies of H-Ras-Fcells .More data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of HRAS (unknown origin) transfected in BALB/c nude mouse incubated for 3 days measured by immunoblot analysisMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of [35S]methionine labelled HRAS in rat Rat1 cells by immunoprecipitation analysisMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Concentration required to inhibit 50% of the cultured colonies of H-Ras-Fcells .More data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Concentration required to inhibit 50% of the cultured colonies of H-Ras-Fcells .More data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Concentration required to inhibit 50% of the cultured colonies of H-Ras-Fcells .More data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Tested for 50% inhibition of generation of Human Ha-ras polymerase chain reaction(PCR) productsMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Concentration required to inhibit 50% of the cultured colonies of H-Ras-Fcells .More data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 310nMAssay Description:Concentration required to inhibit 50% of the cultured colonies of H-Ras-Fcells .More data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Concentration required to inhibit 50% of the cultured colonies of H-Ras-Fcells .More data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Concentration required to inhibit 50% of the cultured colonies of H-Ras-Fcells .More data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Concentration required to inhibit 50% of the cultured colonies of H-Ras-Fcells .More data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 710nMAssay Description:Concentration required to inhibit 50% of the cultured colonies of H-Ras-Fcells .More data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Concentration required to inhibit 50% of the cultured colonies of H-Ras-Fcells .More data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Concentration required to inhibit 50% of the cultured colonies of H-Ras-Fcells .More data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of nucleotide exchange process of oncogenic Ras in vitroMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of nucleotide exchange process of oncogenic Ras in vitroMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 2.55E+3nMAssay Description:Inhibition of human recombinant p21RAS by GDPX assayMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of nucleotide exchange process of oncogenic Ras in vitroMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 4.30E+3nMAssay Description:Concentration required to inhibit 50% of the cultured colonies of H-Ras-Fcells .More data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of nucleotide exchange process of oncogenic Ras in vitroMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of nucleotide exchange process of oncogenic Ras in vitroMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 6.30E+3nMAssay Description:Concentration required to inhibit 50% of the cultured colonies of H-Ras-Fcells .More data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of nucleotide exchange process of oncogenic Ras in vitroMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of nucleotide exchange process of oncogenic Ras in vitroMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of nucleotide exchange process of oncogenic Ras in vitroMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of nucleotide exchange process of oncogenic Ras in vitroMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of Ha-ras polymerase-chain reaction productMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro for inhibition of nucleotide exchange process of oncogenic RasMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of nucleotide exchange process of oncogenic Ras in vitroMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of nucleotide exchange process of oncogenic Ras in vitroMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of nucleotide exchange process of oncogenic Ras in vitroMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of nucleotide exchange process of oncogenic Ras in vitroMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of nucleotide exchange process of oncogenic Ras in vitroMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 1.43E+4nMAssay Description:Concentration required to inhibit 50% of the cultured colonies of H-Ras-Fcells .More data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of nucleotide exchange process of oncogenic Ras in vitroMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of nucleotide exchange process of oncogenic Ras in vitroMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GST-tagged HRAS (1 to 166 residues) (unknown origin) assessed as inhibition of mSOS1 mediated nucleotide exchange by [35S]GTPgammaS bas...More data for this Ligand-Target Pair
Ligand Info
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of nucleotide exchange process of oncogenic Ras in vitroMore data for this Ligand-Target Pair
TargetGTPase HRas(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Massachusetts College Of Pharmacy And Health Sciences University
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of nucleotide exchange process of oncogenic Ras in vitroMore data for this Ligand-Target Pair